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SLB # Authors Title Journal Reference


Martinelli, J.R.; Freckmann, D.M.M.; Buchwald, S.L.

Convenient Method for the Preparation of Weinreb Amides via Pd-Catalyzed Aminocarbonylation of Aryl Bromides at Atmospheric Pressure

Org. Lett. 2006, 8, 4843-4846


Martin, R.; Rodriguez Rivero, M.; Buchwald, S.L.

Domino Copper-Catalyzed C-N coupling-Hydroamidation: A Highly efficient Synthesis of Nitrogen Heterocycles

Angew. Chem., Int. Ed. 2006, 45, 7079-7082


Anderson, K.W.; Ikawa, T.; Tundel, R.E.; Buchwald, S.L

The Selective Reaction of Aryl Halides with KOH: Synthesis of Phenols, Aromatic Ethers and Benzofurans

J. Am. Chem. Soc. 2006, 128, 10694-10695


Anderson, K.W.; Tundel, R.E.; Ikawa, T.; Altman, R.A.; Buchwald, S.L.

Monodentate Phosphines Provide Highly Active Catalysts for Palladium-Catalyzed C-N Bond-Forming Reactions of Heteroaromatic Halides/Amines and (H)N-Heterocycles

Angew. Chem., Int. Ed. 2006, 45, 6523-6527


Shafir, A.; Buchwald, S.L

Highly Selective Room Temperature Copper-Catalyzed C-N Coupling Reactions

J. Am. Chem. Soc. 2006, 128, 8742-8743


Altman, Ryan A.; Buchwald, S.L.

4,7-Dimethoxy-1,10-Phenanthroline: An Excellent Ligand for the Cu-Catalyzed N-Arylation of Imidazoles

Org. Lett. 2006, 8, 2779-2782


Larsen, C.H.; Anderson, K.W.; Tundel, R.E.; Buchwald, S.L.

Palladium-Catalyzed Heck Alkynylation of Benzyl Chlorides

SynLett. 2006, 18, 2941-2946


Burgos, C.H.; Barder, T.E.; Huang, X.; Buchwald, S.L.

Significantly Improved Method for the Palladium-Catalyzed Coupling of Phenols with Aryl Halides:  Understanding Ligand Effects in Phenol/Aryl Halide Coupling Reactions

Angew. Chem. Int. Ed. 2006, 45, 4321-4326


Enguehard-Gueiffier, C.; Thery, I.; Gueiffier, A.; Buchwald, S.L.

A General and Efficient Method for the Copper-catalyzed Cross-coupling of Amides and Thiophenols with 6-Halogenoimidazo[1,2-a]pyridines

Tetrahedron 2006, 62, 6042-6049


Billingsley, K. L.; Anderson, K. W.; Buchwald, S.L.

A Highly Active Catalyst for Suzuki-Miyaura Cross-Coupling Reactions of Heteroaryl Compounds

Angew. Chem., Int. Ed. 2006, 45, 3484-3488


Klingensmith, L.M.; Strieter, E.R.; Barder; Buchwald, S.L.

New Insights into Xantphos/Pd Catalyzed C-N Bond Forming Reactions:  A Structural and Kinetic Study

Organometallics2006, 25, 82-91


Tundel, R.E.; Anderson, K.E.; Buchwald, S. L.

Expedited Palladium-Catalyzed Amination of Aryl Nonaflates Through the Use of Microwave-Irradiation and Soluble Organic Amine Bases

J. Org. Chem. 2006, 71, 430-433


Shekhar, S.; Ryberg, P.; Hartwig, J.F.; Mathew, J.S.; Blackmond, D.G.; Strieter, E.R.; Buchwald, S.L.

A Reevaluation of the Mechanism of the Amination of Aryl Halides Catalyzed by BINAP-Ligated Palladium Complexes

J. Am. Chem. Soc. 2006,128, 3584-3591


Strieter, E.R.; Buchwald, S.L.

Evidence for the Formation and Structure of Palladacycles during Pd-Catalyzed C-N Bond Formation with Catalysts Derived from Bulky Monophosphinobiaryl Ligands

Angew. Chem. Int. Ed.2006, 45, 925-928


Buchwald, S. L.; Mauger, C.; Mignani, G.; Scholz, U.

Industrial-Scale Palladium-Catalyzed Coupling of Aryl Halides and Amines - A Personal Account

Adv. Syn. & Cat. 2006, 348(1+2), 23-39

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SLB # Authors Title Journal Reference


Tsang, W.C.; Zheng, Nan; Buchwald, S. L.

Combined C-H Functionalization/ C-N Bond Formation Route to Carbazoles

J. Am. Chem. Soc. 2005, 127, 14560-14561


Charles, M.D.; Schultz, P.; Buchwald, S. L.

Efficient Pd-Catalyzed Amination of Heteroaryl Halides

Org. Lett. 2005, 7, 3965-3968


Hennessy, E.J.; Buchwald, S. L.

Synthesis of 4,5-Dianilinophthalimide and Related Analogs for Potential Treatment of Alzheimer's Disease via Palladium-Catalyzed Amination

J. Org. Chem. 2005, 70, 7371-7375


Anderson, K.W.; Buchwald, S. L.

General Catalysts for the Suzuki-Miyaura and Sonogashira Coupling Reactions of Aryl Chlorides and for the Coupling of Challenging Substrate Combinations in Water

Angew. Chem., Int. Ed. 2005, 44, 6173-6177


Rainka, M.P.;Milne, J.E.; Buchwald, S. L.

Dynamic Kinetic Resolution of a,b-Unsaturated Lactones Through Asymmetric Copper-Catalyzed Conjugate Reduction: Application to the Total Synthesis of Eupomatilone-3

Angew. Chem., Int. Ed. 2005, 44, 6177-6180


Vorogushin, A.V.; Huang, X.; Buchwald, S. L.

Use of Tunable Ligands Allows for Intermolecular Pd-Catalyzed C-O Bond Formation

J. Am. Chem. Soc. 2005, 127, 8146-8149


Strieter, E.R.; Blackmond, D.I.; Buchwald, S. L.

The Role of Chelating Ligands in the Goldberg Reaction: A Kinetic Study on the Copper-Catalyzed Amidation of Aryl Iodides

J. Am. Chem. Soc. 2005, 127, 4120-4121


Barder, T.E.; Walker, S.D.; Martinelli, J.R.; Buchwald, S. L.

New Catalysts for Suzuki-Miyaura Coupling Processes: Scope and Studies of the Effect of Ligand Structure

J. Am. Chem. Soc. 2005, 127, 4685-4696

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